PDB Information

PDB3JPV
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Synthesis, kinase inhibitory potencies, and in vitro antiproliferative evaluation of new pim kinase inhibitors.
Akue-Gedu, R., Rossignol, E., Azzaro, S., Knapp, S., Filippakopoulos, P., Bullock, A.N., Bain, J., Cohen, P., Prudhomme, M., Anizon, F., Moreau, P.
J.Med.Chem.
HeaderTransferase / Transferase Inhibitor
Released2009-09-04
Resolution2.350
CATH Insert Date01 Nov, 2009

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 01 Nov, 2009 Chopped
B 01 Nov, 2009 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3jpvA01 07 Apr, 2010 3.30.200.20 Assigned
3jpvA02 07 Apr, 2010 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P11309 PIM1_HUMAN Homo sapiens Serine/threonine-protein kinase pim-1