PDB 3itz
PDB Information
| PDB | 3ITZ |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Part 2: Structure-activity relationship (SAR) investigations of fused pyrazoles as potent, selective and orally available inhibitors of p38alpha mitogen-activated protein kinase.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase |
| Released | 2009-08-28 |
| Resolution | 2.250 |
| CATH Insert Date | 04 Mar, 2010 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 05 Mar, 2010 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3itzA01 | 04 Apr, 2010 | 3.30.200.20 | Assigned |
| 3itzA02 | 04 Apr, 2010 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q16539 | MK14_HUMAN | Homo sapiens | Mitogen-activated protein kinase 14 |
