PDB Information

PDB3I7E
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 1
Primary Citation
Design, Synthesis, Protein-Ligand X-ray Structure, and Biological Evaluation of a Series of Novel Macrocyclic Human Immunodeficiency Virus-1 Protease Inhibitors to Combat Drug Resistance.
Ghosh, A.K., Kulkarni, S., Anderson, D.D., Hong, L., Baldridge, A., Wang, Y.F., Chumanevich, A.A., Kovalevsky, A.Y., Tojo, Y., Amano, M., Koh, Y., Tang, J., Weber, I.T., Mitsuya, H.
J.Med.Chem.
HeaderHydrolase
Released2009-07-08
Resolution1.700
CATH Insert Date01 Oct, 2009

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 01 Oct, 2009 Chopped
B 01 Oct, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3i7eA00 14 Mar, 2010 2.40.70.10 Assigned
3i7eB00 14 Mar, 2010 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P03369 POL_HV1A2 HIV-1 M:B_ARV2/SF2 Gag-Pol polyprotein
P03369 POL_HV1A2 HIV-1 M:B_ARV2/SF2 Gag-Pol polyprotein