PDB Information

PDB3HD3
MethodX-RAY DIFFRACTION
Host OrganismPichia pastoris
Gene SourceTrypanosoma cruzi
Primary Citation
Novel non-peptidic vinylsulfones targeting the S2 and S3 subsites of parasite cysteine proteases.
Bryant, C., Kerr, I.D., Debnath, M., Ang, K.K., Ratnam, J., Ferreira, R.S., Jaishankar, P., Zhao, D., Arkin, M.R., McKerrow, J.H., Brinen, L.S., Renslo, A.R.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2009-05-06
Resolution1.750
CATH Insert Date08 Oct, 2009

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 09 Oct, 2009 Chopped
B 09 Oct, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3hd3A00 11 Feb, 2010 3.90.70.10 Assigned
3hd3B00 11 Feb, 2010 3.90.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain