PDB Information

PDB3H0E
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
3,4-Dihydropyrimido(1,2-a)indol-10(2H)-ones as potent non-peptidic inhibitors of caspase-3
Havran, L.M., Chong, D.C., Childers, W.E., Dollings, P.J., Dietrich, A., Harrison, B.L., Marathias, V., Tawa, G., Aulabaugh, A., Cowling, R., Kapoor, B., Xu, W., Mosyak, L., Moy, F., Hum, W.T., Wood, A., Robichaud, A.J.
Bioorg.Med.Chem.
HeaderHydrolase
Released2009-04-09
Resolution2.000
CATH Insert Date26 Nov, 2009

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 26 Nov, 2009 Chopped
B 26 Nov, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3h0eA00 23 Jul, 2010 3.40.50.1460 Assigned
3h0eB00 23 Jul, 2010 3.40.50.1460 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P42574 CASP3_HUMAN Homo sapiens Caspase-3
P42574 CASP3_HUMAN Homo sapiens Caspase-3