PDB Information

PDB3F5X
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
2-(6-Phenyl-1H-indazol-3-yl)-1H-benzo[d]imidazoles: Design and synthesis of a potent and isoform selective PKC-zeta inhibitor.
Trujillo, J.I., Kiefer, J.R., Huang, W., Thorarensen, A., Xing, L., Caspers, N.L., Day, J.E., Mathis, K.J., Kretzmer, K.K., Reitz, B.A., Weinberg, R.A., Stegeman, R.A., Wrightstone, A., Christine, L., Compton, R., Li, X.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Cell Cycle
Released2008-11-04
Resolution2.400
CATH Insert Date05 Feb, 2009

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 05 Feb, 2009 Chopped
B 05 Feb, 2009 Chopped
C 05 Feb, 2009 Chopped
D 05 Feb, 2009 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
3f5xA01 19 Feb, 2009 3.30.200.20 Assigned
3f5xA02 19 Feb, 2009 1.10.510.10 Assigned
3f5xB01 18 Feb, 2009 1.10.472.10 Assigned
3f5xB02 18 Feb, 2009 1.10.472.10 Assigned
3f5xC01 19 Feb, 2009 3.30.200.20 Assigned
3f5xC02 19 Feb, 2009 1.10.510.10 Assigned
3f5xD01 19 Feb, 2009 1.10.472.10 Assigned
3f5xD02 19 Feb, 2009 1.10.472.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2