PDB Information

PDB3ET1
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Scaffold-based discovery of indeglitazar, a PPAR pan-active anti-diabetic agent
Artis, D.R., Lin, J.J., Zhang, C., Wang, W., Mehra, U., Perreault, M., Erbe, D., Krupka, H.I., England, B.P., Arnold, J., Plotnikov, A.N., Marimuthu, A., Nguyen, H., Will, S., Signaevsky, M., Kral, J., Cantwell, J., Settachatgull, C., Yan, D.S., Fong, D., Oh, A., Shi, S., Womack, P., Powell, B., Habets, G., West, B.L., Zhang, K.Y., Milburn, M.V., Vlasuk, G.P., Hirth, K.P., Nolop, K., Bollag, G., Ibrahim, P.N., Tobin, J.F.
Proc.Natl.Acad.Sci.USA
HeaderTranscription/Transferase
Released2008-10-06
Resolution2.500
CATH Insert Date19 Feb, 2009

PDB Images (7)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 19 Feb, 2009 Chopped
B 19 Feb, 2009 Chopped
P 19 Feb, 2009 Rejected
Q 19 Feb, 2009 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3et1A00 21 Mar, 2011 1.10.565.10 Assigned
3et1B00 21 Mar, 2011 1.10.565.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q07869 PPARA_HUMAN Homo sapiens Peroxisome proliferator-activated receptor alpha
Q15788 NCOA1_HUMAN Homo sapiens Nuclear receptor coactivator 1
Q07869 PPARA_HUMAN Homo sapiens Peroxisome proliferator-activated receptor alpha
Q15788 NCOA1_HUMAN Homo sapiens Nuclear receptor coactivator 1