PDB Information

PDB3E8R
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Discovery of novel hydroxamates as highly potent tumor necrosis factor-alpha converting enzyme inhibitors. Part II: optimization of the S3' pocket.
Mazzola, R.D., Zhu, Z., Sinning, L., McKittrick, B., Lavey, B., Spitler, J., Kozlowski, J., Neng-Yang, S., Zhou, G., Guo, Z., Orth, P., Madison, V., Sun, J., Lundell, D., Niu, X.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2008-08-20
Resolution1.900
CATH Insert Date23 Oct, 2008

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 23 Oct, 2008 Chopped
B 23 Oct, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3e8rA00 25 Oct, 2008 3.40.390.10 Assigned
3e8rB00 25 Oct, 2008 3.40.390.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17
P78536 ADA17_HUMAN Homo sapiens Disintegrin and metalloproteinase domain-containing protein 17