PDB Information

PDB3E8C
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceBos taurus
Primary Citation
Aminofurazans as potent inhibitors of AKT kinase
Rouse, M.B., Seefeld, M.A., Leber, J.D., McNulty, K.C., Sun, L., Miller, W.H., Zhang, S., Minthorn, E.A., Concha, N.O., Choudhry, A.E., Schaber, M.D., Heerding, D.A.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-08-19
Resolution2.200
CATH Insert Date20 Nov, 2008

PDB Images (25)

PDB Prints

PDB Chains (12)

Chain ID Date inserted into CATH CATH Status
A 20 Nov, 2008 Chopped
B 20 Nov, 2008 Chopped
C 20 Nov, 2008 Chopped
D 20 Nov, 2008 Chopped
E 20 Nov, 2008 Chopped
F 20 Nov, 2008 Chopped
G 20 Nov, 2008 Rejected
H 20 Nov, 2008 Rejected
I 20 Nov, 2008 Rejected
J 20 Nov, 2008 Rejected
K 20 Nov, 2008 Rejected
L 20 Nov, 2008 Rejected

CATH Domains (12)

Domain ID Date inserted into CATH Superfamily CATH Status
3e8cA01 08 Dec, 2008 1.10.510.10 Assigned
3e8cA02 08 Dec, 2008 3.30.200.20 Assigned
3e8cB01 08 Dec, 2008 1.10.510.10 Assigned
3e8cB02 08 Dec, 2008 3.30.200.20 Assigned
3e8cC01 08 Dec, 2008 1.10.510.10 Assigned
3e8cC02 08 Dec, 2008 3.30.200.20 Assigned
3e8cD01 08 Dec, 2008 1.10.510.10 Assigned
3e8cD02 08 Dec, 2008 3.30.200.20 Assigned
3e8cE01 08 Dec, 2008 1.10.510.10 Assigned
3e8cE02 08 Dec, 2008 3.30.200.20 Assigned
3e8cF01 08 Dec, 2008 1.10.510.10 Assigned
3e8cF02 08 Dec, 2008 3.30.200.20 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha