PDB Information

PDB3CXW
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
7,8-Dichloro-1-oxo-beta-carbolines as a Versatile Scaffold for the Development of Potent and Selective Kinase Inhibitors with Unusual Binding Modes
Huber, K., Brault, L., Fedorov, O., Gasser, C., Filippakopoulos, P., Bullock, A.N., Fabbro, D., Trappe, J., Schwaller, J., Knapp, S., Bracher, F.
J.Med.Chem.
HeaderTransferase
Released2008-04-25
Resolution2.100
CATH Insert Date23 Jul, 2008

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 24 Jul, 2008 Chopped
B 24 Jul, 2008 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3cxwA01 26 Jul, 2008 3.30.200.20 Assigned
3cxwA02 26 Jul, 2008 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P11309 PIM1_HUMAN Homo sapiens Serine/threonine-protein kinase pim-1