PDB Information

PDB3CPB
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Discovery of Aryl Aminoquinazoline Pyridones as Potent, Selective, and Orally Efficacious Inhibitors of Receptor Tyrosine Kinase c-Kit.
Hu, E., Tasker, A., White, R.D., Kunz, R.K., Human, J., Chen, N., Burli, R., Hungate, R., Novak, P., Itano, A., Zhang, X., Yu, V., Nguyen, Y., Tudor, Y., Plant, M., Flynn, S., Xu, Y., Meagher, K.L., Whittington, D.A., Ng, G.Y.
J.Med.Chem.
HeaderTransferase
Released2008-03-31
Resolution2.700
CATH Insert Date23 Jul, 2008

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 24 Jul, 2008 Chopped
B 24 Jul, 2008 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3cpbA01 10 Sep, 2008 3.30.200.20 Assigned
3cpbA02 10 Sep, 2008 1.10.510.10 Assigned
3cpbB01 10 Sep, 2008 3.30.200.20 Assigned
3cpbB02 10 Sep, 2008 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P35968 VGFR2_HUMAN Homo sapiens Vascular endothelial growth factor receptor 2
P35968 VGFR2_HUMAN Homo sapiens Vascular endothelial growth factor receptor 2