PDB Information

PDB3CLD
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
X-ray crystal structure of the novel enhanced-affinity glucocorticoid agonist fluticasone furoate in the glucocorticoid receptor-ligand binding domain.
Biggadike, K., Bledsoe, R.K., Hassell, A.M., Kirk, B.E., McLay, I.M., Shewchuk, L.M., Stewart, E.L.
J.Med.Chem.
HeaderTranscription
Released2008-03-18
Resolution2.840
CATH Insert Date23 Jul, 2008

PDB Images (7)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 24 Jul, 2008 Chopped
B 24 Jul, 2008 Chopped
C 24 Jul, 2008 Rejected
H 24 Jul, 2008 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3cldA00 25 Jul, 2008 1.10.565.10 Assigned
3cldB00 25 Jul, 2008 1.10.565.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2