PDB Information

PDB3BE2
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Naphthamides as novel and potent vascular endothelial growth factor receptor tyrosine kinase inhibitors: design, synthesis, and evaluation.
Harmange, J.C., Weiss, M.M., Germain, J., Polverino, A.J., Borg, G., Bready, J., Chen, D., Choquette, D., Coxon, A., Demelfi, T., Dipietro, L., Doerr, N., Estrada, J., Flynn, J., Graceffa, R.F., Harriman, S.P., Kaufman, S., La, D.S., Long, A., Martin, M.W., Neervannan, S., Patel, V.F., Potashman, M., Regal, K., Roveto, P.M., Schrag, M.L., Starnes, C., Tasker, A., Teffera, Y., Wang, L., White, R.D., Whittington, D.A., Zanon, R.
J.Med.Chem.
HeaderTransferase
Released2007-11-16
Resolution1.750
CATH Insert Date10 Apr, 2008

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 10 Apr, 2008 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3be2A01 10 Sep, 2008 3.30.200.20 Assigned
3be2A02 10 Sep, 2008 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P35968 VGFR2_HUMAN Homo sapiens Vascular endothelial growth factor receptor 2