PDB Information

PDB3B8R
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Evaluation of a Series of Naphthamides as Potent, Orally Active Vascular Endothelial Growth Factor Receptor-2 Tyrosine Kinase Inhibitors
Weiss, M.M., Harmange, J.C., Polverino, A.J., Bauer, D., Berry, L., Berry, V., Borg, G., Bready, J., Chen, D., Choquette, D., Coxon, A., DeMelfi, T., Doerr, N., Estrada, J., Flynn, J., Graceffa, R.F., Harriman, S.P., Kaufman, S., La, D.S., Long, A., Neervannan, S., Patel, V.F., Potashman, M., Regal, K., Roveto, P.M., Schrag, M.L., Starnes, C., Tasker, A., Teffera, Y., Whittington, D.A., Zanon, R.
J.Med.Chem.
HeaderTransferase
Released2007-11-01
Resolution2.700
CATH Insert Date03 Apr, 2008

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Apr, 2008 Chopped
B 03 Apr, 2008 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3b8rA01 10 Sep, 2008 3.30.200.20 Assigned
3b8rA02 10 Sep, 2008 1.10.510.10 Assigned
3b8rB01 10 Sep, 2008 3.30.200.20 Assigned
3b8rB02 10 Sep, 2008 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P35968 VGFR2_HUMAN Homo sapiens Vascular endothelial growth factor receptor 2
P35968 VGFR2_HUMAN Homo sapiens Vascular endothelial growth factor receptor 2