PDB Information

PDB2ZIS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
Synthesis and structure-activity relationships of novel benzofuran farnesyltransferase inhibitors
Asoh, K., Kohchi, M., Hyoudoh, I., Ohtsuka, T., Masubuchi, M., Kawasaki, K., Ebiike, H., Shiratori, Y., Fukami, T.A., Kondoh, O., Tsukaguchi, T., Ishii, N., Aoki, Y., Shimma, N., Sakaitani, M.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2008-02-22
Resolution2.600
CATH Insert Date26 Feb, 2009

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 26 Feb, 2009 Chopped
B 26 Feb, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2zisA00 03 Mar, 2009 1.25.40.120 Assigned
2zisB00 03 Mar, 2009 1.50.10.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q02293 FNTB_RAT Rattus norvegicus Protein farnesyltransferase subunit beta
Q04631 FNTA_RAT Rattus norvegicus Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha