PDB Information

PDB2VNY
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceBOS TAURUS
Primary Citation
Identification of 4-(4-Aminopiperidin-1-Yl)-7H-Pyrrolo[2,3-D]Pyrimidines as Selective Inhibitors of Protein Kinase B Through Fragment Elaboration.
Caldwell, J.J., Davies, T.G., Donald, A., Mchardy, T., Rowlands, M.G., Aherne, G.W., Hunter, L.K., Taylor, K., Ruddle, R., Raynaud, F.I., Verdonk, M., Workman, P., Garrett, M.D., Collins, I.
J.Med.Chem.
HeaderTransferase
Released2008-02-08
Resolution1.960
CATH Insert Date10 Apr, 2008

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 10 Apr, 2008 Chopped
I 10 Apr, 2008 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2vnyA01 08 Dec, 2008 1.10.510.10 Assigned
2vnyA02 08 Dec, 2008 3.30.200.20 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P00517 KAPCA_BOVIN Bos taurus cAMP-dependent protein kinase catalytic subunit alpha