PDB Information

PDB2VNT
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Selective Urokinase-Type Plasminogen Activator (Upa) Inhibitors 4. 1-(7-Sulphonamidoisoquinolinyl) Guanidines
Fish, P.V., Barber, C.G., Brown, D.G., Butt, R., Henry, B.T., Horne, V., Huggins, J.P., Mccleverty, D., Phillips, C., Webster, R., Dickinson, R.P., Collis, M.G., King, E., O'Gara, M., Mcintosh, F.
J.Med.Chem.
HeaderHydrolase
Released2008-02-07
Resolution2.200
CATH Insert Date21 Feb, 2008

PDB Images (19)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 21 Feb, 2008 Chopped
B 21 Feb, 2008 Chopped
C 21 Feb, 2008 Chopped
D 21 Feb, 2008 Chopped
E 21 Feb, 2008 Chopped
F 21 Feb, 2008 Chopped

CATH Domains (12)

Domain ID Date inserted into CATH Superfamily CATH Status
2vntA01 23 Feb, 2008 2.40.10.10 Assigned
2vntA02 23 Feb, 2008 2.40.10.10 Assigned
2vntB01 23 Feb, 2008 2.40.10.10 Assigned
2vntB02 23 Feb, 2008 2.40.10.10 Assigned
2vntC01 23 Feb, 2008 2.40.10.10 Assigned
2vntC02 23 Feb, 2008 2.40.10.10 Assigned
2vntD01 23 Feb, 2008 2.40.10.10 Assigned
2vntD02 23 Feb, 2008 2.40.10.10 Assigned
2vntE01 23 Feb, 2008 2.40.10.10 Assigned
2vntE02 23 Feb, 2008 2.40.10.10 Assigned
2vntF01 23 Feb, 2008 2.40.10.10 Assigned
2vntF02 23 Feb, 2008 2.40.10.10 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P00749 UROK_HUMAN Homo sapiens Urokinase-type plasminogen activator
P00749 UROK_HUMAN Homo sapiens Urokinase-type plasminogen activator
P00749 UROK_HUMAN Homo sapiens Urokinase-type plasminogen activator
P00749 UROK_HUMAN Homo sapiens Urokinase-type plasminogen activator
P00749 UROK_HUMAN Homo sapiens Urokinase-type plasminogen activator
P00749 UROK_HUMAN Homo sapiens Urokinase-type plasminogen activator