PDB Information

PDB2VH0
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Structure and property based design of factor Xa inhibitors: biaryl pyrrolidin-2-ones incorporating basic heterocyclic motifs.
Young, R.J., Borthwick, A.D., Brown, D., Burns-Kurtis, C.L., Campbell, M., Chan, C., Charbaut, M., Convery, M.A., Diallo, H., Hortense, E., Irving, W.R., Kelly, H.A., King, N.P., Kleanthous, S., Mason, A.M., Pateman, A.J., Patikis, A.N., Pinto, I.L., Pollard, D.R., Senger, S., Shah, G.P., Toomey, J.R., Watson, N.S., Weston, H.E., Zhou, P.
Bioorg. Med. Chem. Lett.
HeaderHydrolase
Released2007-11-16
Resolution1.700
CATH Insert Date27 Nov, 2008

PDB Images (6)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 27 Nov, 2008 Chopped
B 27 Nov, 2008 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
2vh0A01 28 Nov, 2008 2.40.10.10 Assigned
2vh0A02 28 Nov, 2008 2.40.10.10 Assigned
2vh0B00 28 Nov, 2008 2.10.25.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00742 FA10_HUMAN Homo sapiens Coagulation factor X
P00742 FA10_HUMAN Homo sapiens Coagulation factor X