PDB 2rgu

PDB Links
Overview

PDB Information

PDB	2RGU
Method	X-RAY DIFFRACTION
Host Organism	Pichia pastoris
Gene Source	Homo sapiens
Primary Citation	8-(3-(R)-Aminopiperidin-1-yl)-7-but-2-ynyl-3-methyl-1-(4-methyl-quinazolin-2-ylmethyl)-3,7-dihydropurine-2,6-dione (BI 1356), a Highly Potent, Selective, Long-Acting, and Orally Bioavailable DPP-4 Inhibitor for the Treatment of Type 2 Diabetes. Eckhardt, M., Langkopf, E., Mark, M., Tadayyon, M., Thomas, L., Nar, H., Pfrengle, W., Guth, B., Lotz, R., Sieger, P., Fuchs, H., Himmelsbach, F. J.Med.Chem.
Header	Hydrolase
Released	2007-10-05
Resolution	2.600
CATH Insert Date	08 Nov, 2007

PDB Images (7)

Image of CATH 2rgu

2rgu

PDB 2rgu

Image of CATH 2rguA

2rguA

PDB Chain 2rguA

Image of CATH 2rguB

2rguB

PDB Chain 2rguB

Image of CATH 2rguA01

2rguA01

CATH Domain 2rguA01

Image of CATH 2rguA02

2rguA02

CATH Domain 2rguA02

Image of CATH 2rguB01

2rguB01

CATH Domain 2rguB01

Image of CATH 2rguB02

2rguB02

CATH Domain 2rguB02

PDB Prints

PDB Chains (2)

Chain ID	Date inserted into CATH	CATH Status
A	08 Nov, 2007	Chopped
B	08 Nov, 2007	Chopped

CATH Domains (4)

Domain ID	Date inserted into CATH	Superfamily	CATH Status
2rguA01	23 Nov, 2007	2.140.10.30	Assigned
2rguA02	23 Nov, 2007	3.40.50.1820	Assigned
2rguB01	23 Nov, 2007	2.140.10.30	Assigned
2rguB02	23 Nov, 2007	3.40.50.1820	Assigned

UniProtKB Entries (2)

Accession	Gene ID	Taxon	Description
P27487	DPP4_HUMAN	Homo sapiens	Dipeptidyl peptidase 4
P27487	DPP4_HUMAN	Homo sapiens	Dipeptidyl peptidase 4