PDB Information

PDB2QT9
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
4-Arylcyclohexylalanine analogs as potent, selective, and orally active inhibitors of dipeptidyl peptidase IV.
Kaelin, D.E., Smenton, A.L., Eiermann, G.J., He, H., Leiting, B., Lyons, K.A., Patel, R.A., Patel, S.B., Petrov, A., Scapin, G., Wu, J.K., Thornberry, N.A., Weber, A.E., Duffy, J.L.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2007-08-01
Resolution2.100
CATH Insert Date08 Nov, 2007

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 Nov, 2007 Chopped
B 08 Nov, 2007 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
2qt9A01 23 Nov, 2007 3.40.50.1820 Assigned
2qt9A02 23 Nov, 2007 2.140.10.30 Assigned
2qt9B01 23 Nov, 2007 3.40.50.1820 Assigned
2qt9B02 23 Nov, 2007 2.140.10.30 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4