PDB 2q8i
PDB Information
| PDB | 2Q8I |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21 |
| Gene Source | Homo sapiens |
| Primary Citation | Distinct Structural Mechanisms for Inhibition of Pyruvate Dehydrogenase Kinase Isoforms by AZD7545, Dichloroacetate, and Radicicol.
Structure
|
| Header | Transferase |
| Released | 2007-06-10 |
| Resolution | 2.600 |
| CATH Insert Date | 26 Jul, 2007 |
PDB Images (6)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 26 Jul, 2007 | Chopped |
| B | 26 Jul, 2007 | Chopped |
CATH Domains (3)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 2q8iA01 | 17 Aug, 2007 | 1.20.140.20 | Assigned |
| 2q8iA02 | 17 Aug, 2007 | 3.30.565.10 | Assigned |
| 2q8iB00 | 16 Aug, 2007 | 2.40.50.100 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P10515 | ODP2_HUMAN | Homo sapiens | Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, mitochondrial |
| Q15120 | PDK3_HUMAN | Homo sapiens | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial |
