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PDB Information
| PDB | 2Q8F |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21 |
| Gene Source | Homo sapiens |
| Primary Citation |
Distinct Structural Mechanisms for Inhibition of Pyruvate Dehydrogenase Kinase Isoforms by AZD7545, Dichloroacetate, and Radicicol.
Kato, M., Li, J., Chuang, J.L., Chuang, D.T.
Structure
|
| Header | Transferase |
| Released | 2007-06-10 |
| Resolution | 2.030 |
| CATH Insert Date | 26 Jul, 2007 |
PDB Images (4)
2q8fA01
CATH Domain 2q8fA01
2q8fA02
CATH Domain 2q8fA02
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
| A | 26 Jul, 2007 | Chopped
|
CATH Domains (2)
UniProtKB Entries (1)
| Accession |
Gene ID |
Taxon |
Description |
| Q15118 |
PDK1_HUMAN |
Homo sapiens |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |