PDB 2q11
PDB Information
PDB | 2Q11 |
Method | X-RAY DIFFRACTION |
Host Organism | unidentified baculovirus |
Gene Source | Homo sapiens |
Primary Citation | 2-Amino-3,4-dihydroquinazolines as inhibitors of BACE-1 (beta-Site APP cleaving enzyme): Use of structure based design to convert a micromolar hit into a nanomolar lead.
J.Med.Chem.
|
Header | Hydrolase |
Released | 2007-05-23 |
Resolution | 2.400 |
CATH Insert Date | 07 Nov, 2007 |
PDB Images (10)
PDB Prints
PDB Chains (3)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 08 Nov, 2007 | Chopped |
B | 08 Nov, 2007 | Chopped |
C | 08 Nov, 2007 | Chopped |
CATH Domains (6)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
2q11A01 | 23 Nov, 2007 | 2.40.70.10 | Assigned |
2q11A02 | 23 Nov, 2007 | 2.40.70.10 | Assigned |
2q11B01 | 23 Nov, 2007 | 2.40.70.10 | Assigned |
2q11B02 | 23 Nov, 2007 | 2.40.70.10 | Assigned |
2q11C01 | 23 Nov, 2007 | 2.40.70.10 | Assigned |
2q11C02 | 23 Nov, 2007 | 2.40.70.10 | Assigned |
UniProtKB Entries (3)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P56817 | BACE1_HUMAN | Homo sapiens | Beta-secretase 1 |
P56817 | BACE1_HUMAN | Homo sapiens | Beta-secretase 1 |
P56817 | BACE1_HUMAN | Homo sapiens | Beta-secretase 1 |