PDB Information

PDB2GA2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Development of sulfonamide compounds as potent methionine aminopeptidase type II inhibitors with antiproliferative properties.
Kawai, M., BaMaung, N.Y., Fidanze, S.D., Erickson, S.A., Tedrow, J.S., Sanders, W.J., Vasudevan, A., Park, C., Hutchins, C., Comess, K.M., Kalvin, D., Wang, J., Zhang, Q., Lou, P., Tucker-Garcia, L., Bouska, J., Bell, R.L., Lesniewski, R., Henkin, J., Sheppard, G.S.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2006-03-07
Resolution1.950
CATH Insert Date15 Mar, 2007

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 15 Mar, 2007 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2ga2A01 24 Jan, 2013 3.90.230.10 Assigned
2ga2A02 24 Jan, 2013 1.10.10.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P50579 MAP2_HUMAN Homo sapiens Methionine aminopeptidase 2