PDB 2g1q
PDB Information
PDB | 2G1Q |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli BL21 |
Gene Source | Homo sapiens |
Primary Citation | Kinesin spindle protein (KSP) inhibitors. Part 4: Structure-based design of 5-alkylamino-3,5-diaryl-4,5-dihydropyrazoles as potent, water-soluble inhibitors of the mitotic kinesin KSP.
Bioorg.Med.Chem.Lett.
|
Header | Cell Cycle |
Released | 2006-02-14 |
Resolution | 2.510 |
CATH Insert Date | 05 Oct, 2006 |
PDB Images (5)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 05 Oct, 2006 | Chopped |
B | 05 Oct, 2006 | Chopped |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
2g1qA00 | 15 Oct, 2006 | 3.40.850.10 | Assigned |
2g1qB00 | 02 Nov, 2006 | 3.40.850.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P52732 | KIF11_HUMAN | Homo sapiens | Kinesin-like protein KIF11 |
P52732 | KIF11_HUMAN | Homo sapiens | Kinesin-like protein KIF11 |