PDB Information

PDB2G0H
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Structure-Based Drug Design of a Novel Family of PPARgamma Partial Agonists: Virtual Screening, X-ray Crystallography, and in Vitro/in Vivo Biological Activities
Lu, I.L., Huang, C.F., Peng, Y.H., Lin, Y.T., Hsieh, H.P., Chen, C.T., Lien, T.W., Lee, H.J., Mahindroo, N., Prakash, E., Yueh, A., Chen, H.Y., Goparaju, C.M., Chen, X., Liao, C.C., Chao, Y.S., Hsu, J.T., Wu, S.Y.
J.Med.Chem.
HeaderTranscription Activator
Released2006-02-13
Resolution2.300
CATH Insert Date14 Jul, 2006

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Jul, 2006 Chopped
B 14 Jul, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
2g0hA00 16 Oct, 2006 1.10.565.10 Assigned
2g0hB00 16 Oct, 2006 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P37231 PPARG_HUMAN Homo sapiens Peroxisome proliferator-activated receptor gamma
P37231 PPARG_HUMAN Homo sapiens Peroxisome proliferator-activated receptor gamma