PDB Information

PDB2G00
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Discovery of potent, efficacious, and orally bioavailable inhibitors of blood coagulation factor Xa with neutral P1 moieties.
Pinto, D.J., Galemmo, R.A., Quan, M.L., Orwat, M.J., Clark, C., Li, R., Wells, B., Woerner, F., Alexander, R.S., Rossi, K.A., Smallwood, A., Wong, P.C., Luettgen, J.M., Rendina, A.R., Knabb, R.M., He, K., Wexler, R.R., Lam, P.Y.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2006-02-10
Resolution2.100
CATH Insert Date05 Oct, 2006

PDB Images (6)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Oct, 2006 Chopped
L 05 Oct, 2006 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
2g00A01 19 Oct, 2006 2.40.10.10 Assigned
2g00A02 19 Oct, 2006 2.40.10.10 Assigned
2g00L00 16 Oct, 2006 2.10.25.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00742 FA10_HUMAN Homo sapiens Coagulation factor X
P00742 FA10_HUMAN Homo sapiens Coagulation factor X