PDB 2e9n
PDB Information
| PDB | 2E9N |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of 1,4-dihydroindeno[1,2-c]pyrazoles as a novel class of potent and selective checkpoint kinase 1 inhibitors.
Bioorg.Med.Chem.
|
| Header | Transferase |
| Released | 2007-01-26 |
| Resolution | 2.500 |
| CATH Insert Date | 21 Feb, 2008 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 21 Feb, 2008 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 2e9nA01 | 23 Feb, 2008 | 3.30.200.20 | Assigned |
| 2e9nA02 | 23 Feb, 2008 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O14757 | CHK1_HUMAN | Homo sapiens | Serine/threonine-protein kinase Chk1 |
