PDB Information

PDB2C0O
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHOMO SAPIENS
Primary Citation
Discovery of A-770041, a Src-Family Selective Orally Active Lck Inhibitor that Prevents Organ Allograft Rejection.
Burchat, A., Borhani, D.W., Calderwood, D.J., Hirst, G.C., Li, B., Stachlewitz, R.F.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2005-09-06
Resolution2.850
CATH Insert Date28 Sep, 2006

PDB Images (11)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 28 Sep, 2006 Chopped
B 28 Sep, 2006 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
2c0oA01 22 Dec, 2006 2.30.30.40 Assigned
2c0oA02 22 Dec, 2006 3.30.505.10 Assigned
2c0oA03 22 Dec, 2006 3.30.200.20 Assigned
2c0oA04 22 Dec, 2006 1.10.510.10 Assigned
2c0oB01 22 Dec, 2006 2.30.30.40 Assigned
2c0oB02 22 Dec, 2006 3.30.505.10 Assigned
2c0oB03 22 Dec, 2006 3.30.200.20 Assigned
2c0oB04 22 Dec, 2006 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P08631 HCK_HUMAN Homo sapiens Tyrosine-protein kinase HCK
P08631 HCK_HUMAN Homo sapiens Tyrosine-protein kinase HCK