PDB 1zkn
PDB Information
| PDB | 1ZKN |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21 |
| Gene Source | Homo sapiens |
| Primary Citation | Crystal Structures of Phosphodiesterases 4 and 5 in Complex with Inhibitor 3-Isobutyl-1-Methylxanthine Suggest a Conformation Determinant of Inhibitor Selectivity
J.Biol.Chem.
|
| Header | Hydrolase |
| Released | 2005-05-03 |
| Resolution | 2.100 |
| CATH Insert Date | 05 Mar, 2006 |
PDB Images (9)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 05 Mar, 2006 | Chopped |
| B | 05 Mar, 2006 | Chopped |
| C | 05 Mar, 2006 | Chopped |
| D | 05 Mar, 2006 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 1zknA00 | 10 Mar, 2006 | 1.10.1300.10 | Assigned |
| 1zknB00 | 10 Mar, 2006 | 1.10.1300.10 | Assigned |
| 1zknC00 | 10 Mar, 2006 | 1.10.1300.10 | Assigned |
| 1zknD00 | 10 Mar, 2006 | 1.10.1300.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q08499 | PDE4D_HUMAN | Homo sapiens | cAMP-specific 3',5'-cyclic phosphodiesterase 4D |
| Q08499 | PDE4D_HUMAN | Homo sapiens | cAMP-specific 3',5'-cyclic phosphodiesterase 4D |
| Q08499 | PDE4D_HUMAN | Homo sapiens | cAMP-specific 3',5'-cyclic phosphodiesterase 4D |
| Q08499 | PDE4D_HUMAN | Homo sapiens | cAMP-specific 3',5'-cyclic phosphodiesterase 4D |
