PDB Information

PDB1YRS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Kinesin spindle protein (KSP) inhibitors. Part 1: The discovery of 3,5-diaryl-4,5-dihydropyrazoles as potent and selective inhibitors of the mitotic kinesin KSP
Cox, C.D., Breslin, M.J., Mariano, B.J., Coleman, P.J., Buser, C.A., Walsh, E.S., Hamilton, K., Huber, H.E., Kohl, N.E., Torrent, M., Yan, Y., Kuo, L.C., Hartman, G.D.
BIOORG.MED.CHEM.LETT.
HeaderCell Cycle
Released2005-02-04
Resolution2.500
CATH Insert Date05 Mar, 2006

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
1yrsA00 10 Mar, 2006 3.40.850.10 Assigned
1yrsB00 10 Mar, 2006 3.40.850.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P52732 KIF11_HUMAN Homo sapiens Kinesin-like protein KIF11
P52732 KIF11_HUMAN Homo sapiens Kinesin-like protein KIF11