PDB Information

PDB1Y8J
MethodX-RAY DIFFRACTION
Host OrganismSaccharomyces cerevisiae
Gene SourceHomo sapiens
Primary Citation
Second-Generation Inhibitors for the Metalloprotease Neprilysin Based on Bicyclic Heteroaromatic Scaffolds: Synthesis, Biological Activity, and X-ray Crystal Structure Analysis
Sahli, S., Frank, B., Schweizer, W.B., Diederich, F., Blum-Kaelin, D., Aebi, J.D., Bohm, H.J., Oefner, C., Dale, G.E.
HELV.CHIM.ACTA
HeaderHydrolase
Released2004-12-13
Resolution2.250
CATH Insert Date05 Mar, 2006

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
1y8jA01 09 Mar, 2006 3.40.390.10 Assigned
1y8jA02 09 Mar, 2006 1.10.1380.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P08473 NEP_HUMAN Homo sapiens Neprilysin