PDB Information

PDB1XGJ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli K12
Gene SourceEscherichia coli
Primary Citation
Structure-based optimization of a non-beta-lactam lead results in inhibitors that do not up-regulate beta-lactamase expression in cell culture.
Tondi, D., Morandi, F., Bonnet, R., Costi, M.P., Shoichet, B.K.
J.Am.Chem.Soc.
HeaderHydrolase
Released2004-09-17
Resolution1.970
CATH Insert Date05 Mar, 2006

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
1xgjA00 09 Mar, 2006 3.40.710.10 Assigned
1xgjB00 09 Mar, 2006 3.40.710.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00811 AMPC_ECOLI Escherichia coli K-12 Beta-lactamase
P00811 AMPC_ECOLI Escherichia coli K-12 Beta-lactamase