PDB 1x81
PDB Information
| PDB | 1X81 |
| Method | X-RAY DIFFRACTION |
| Host Organism | |
| Gene Source | |
| Primary Citation | Design, synthesis, and activity of 4-quinolone and pyridone compounds as nonthiol-containing farnesyltransferase inhibitors.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase |
| Released | 2004-08-16 |
| Resolution | 3.500 |
| CATH Insert Date | 05 Mar, 2006 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 05 Mar, 2006 | Chopped |
| B | 05 Mar, 2006 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 1x81A00 | 09 Mar, 2006 | 1.25.40.120 | Assigned |
| 1x81B00 | 09 Mar, 2006 | 1.50.10.20 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q04631 | FNTA_RAT | Rattus norvegicus | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha |
| Q02293 | FNTB_RAT | Rattus norvegicus | Protein farnesyltransferase subunit beta |
