PDB 1wok
PDB Information
| PDB | 1WOK |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of quinazolinone and quinoxaline derivatives as potent and selective poly(ADP-ribose) polymerase-1/2 inhibitors.
Febs Lett.
|
| Header | Transferase |
| Released | 2004-08-20 |
| Resolution | 3.000 |
| CATH Insert Date | 05 Mar, 2006 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 05 Mar, 2006 | Chopped |
| B | 05 Mar, 2006 | Chopped |
| C | 05 Mar, 2006 | Chopped |
| D | 05 Mar, 2006 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 1wokA01 | 09 Mar, 2006 | 1.20.142.10 | Assigned |
| 1wokA02 | 09 Mar, 2006 | 3.90.228.10 | Assigned |
| 1wokB01 | 09 Mar, 2006 | 1.20.142.10 | Assigned |
| 1wokB02 | 09 Mar, 2006 | 3.90.228.10 | Assigned |
| 1wokC01 | 09 Mar, 2006 | 1.20.142.10 | Assigned |
| 1wokC02 | 09 Mar, 2006 | 3.90.228.10 | Assigned |
| 1wokD01 | 09 Mar, 2006 | 1.20.142.10 | Assigned |
| 1wokD02 | 09 Mar, 2006 | 3.90.228.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P09874 | PARP1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase 1 |
| P09874 | PARP1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase 1 |
| P09874 | PARP1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase 1 |
| P09874 | PARP1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase 1 |
