PDB Information

PDB1VSN
MethodX-RAY DIFFRACTION
Host OrganismPichia pastoris
Gene SourceHomo sapiens
Primary Citation
Identification of a potent and selective non-basic cathepsin K inhibitor.
Li, C.S., Deschenes, D., Desmarais, S., Falgueyret, J.P., Gauthier, J.Y., Kimmel, D.B., McGrath, M.E., McKay, D.J., Percival, M.D., Riendeau, D., Rodan, S.B., Truong, V.L., Wesolowski, G., Zamboni, R., Black, W.C.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2007-03-19
Resolution2.000
CATH Insert Date26 Apr, 2007

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 26 Apr, 2007 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
1vsnA00 29 Jul, 2008 3.90.70.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P43235 CATK_HUMAN Homo sapiens Cathepsin K