PDB Information

PDB1U65
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
The crystal structure of the complex of the anticancer prodrug 7-ethyl-10-[4-(1-piperidino)-1-piperidino]-carbonyloxycamptothecin (CPT-11) with Torpedo californica acetylcholinesterase provides a molecular explanation for its cholinergic action
Harel, M., Hyatt, J.L., Brumshtein, B., Morton, C.L., Yoon, K.J., Wadkins, R.M., Silman, I., Sussman, J.L., Potter, P.M.
Mol.Pharmacol.
HeaderHydrolase
Released2004-07-29
Resolution2.610
CATH Insert Date05 Mar, 2006

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
1u65A00 09 Mar, 2006 3.40.50.1820 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P04058 ACES_TETCF Tetronarce californica Acetylcholinesterase