PDB Information

PDB1U3R
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Design and synthesis of aryl diphenolic azoles as potent and selective estrogen receptor-beta ligands.
Malamas, M.S., Manas, E.S., McDevitt, R.E., Gunawan, I., Xu, Z.B., Collini, M.D., Miller, C.P., Dinh, T., Henderson, R.A., Keith Jr., J.C., Harris, H.A.
J.Med.Chem.
HeaderTranscription
Released2004-07-22
Resolution2.210
CATH Insert Date05 Mar, 2006

PDB Images (7)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped
C 05 Mar, 2006 Rejected
D 05 Mar, 2006 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
1u3rA00 09 Mar, 2006 1.10.565.10 Assigned
1u3rB00 09 Mar, 2006 1.10.565.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q92731 ESR2_HUMAN Homo sapiens Estrogen receptor beta
Q15788 NCOA1_HUMAN Homo sapiens Nuclear receptor coactivator 1
Q15788 NCOA1_HUMAN Homo sapiens Nuclear receptor coactivator 1
Q92731 ESR2_HUMAN Homo sapiens Estrogen receptor beta