PDB Information

PDB1RDT
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Structure-based design of potent retinoid X receptor alpha agonists.
Haffner, C.D., Lenhard, J.M., Miller, A.B., McDougald, D.L., Dwornik, K., Ittoop, O.R., Gampe Jr., R.T., Xu, H.E., Blanchard, S., Montana, V.G., Consler, T.G., Bledsoe, R.K., Ayscue, A., Croom, D.
J.Med.Chem.
HeaderHormone/Growth Factor
Released2003-11-06
Resolution2.400
CATH Insert Date05 Mar, 2006

PDB Images (7)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Rejected
D 05 Mar, 2006 Chopped
E 05 Mar, 2006 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
1rdtA00 05 Mar, 2006 1.10.565.10 Assigned
1rdtD00 05 Mar, 2006 1.10.565.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q15788 NCOA1_HUMAN Homo sapiens Nuclear receptor coactivator 1
P19793 RXRA_HUMAN Homo sapiens Retinoic acid receptor RXR-alpha
Q92793 CBP_HUMAN Homo sapiens CREB-binding protein
P37231 PPARG_HUMAN Homo sapiens Peroxisome proliferator-activated receptor gamma