PDB Information

PDB1PYE
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
The discovery of a new structural class of cyclin-dependent kinase inhibitors, aminoimidazo[1,2-a]pyridines.
Hamdouchi, C., Keyser, H., Collins, E., Jaramillo, C., De Diego, J.E., Spencer, C.D., Dempsey, J.A., Anderson, B.D., Leggett, T., Stamm, N.B., Schultz, R.M., Watkins, S.A., Cocke, K., Lemke, S., Burke, T.F., Beckmann, R.P., Dixon, J.T., Gurganus, T.M., Rankl, N.B., Houck, K.A., Zhang, F., Vieth, M., Espinosa, J., Timm, D.E., Campbell, R.M., Patel, B.K., Brooks, H.B.
MOL.CANCER THER.
HeaderTransferase
Released2003-07-08
Resolution2.000
CATH Insert Date05 Mar, 2006

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
1pyeA01 05 Mar, 2006 3.30.200.20 Assigned
1pyeA02 05 Mar, 2006 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2