PDB Information

PDB1NLJ
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Azepanone-Based Inhibitors of Human and Rat Cathepsin K
Marquis, R.W., Ru, Y., LoCastro, S.M., Zeng, J., Yamashita, D.S., Oh, H.J., Erhard, K.F., Davis, L.D., Tomaszek, T.A., Tew, D., Salyers, K., Proksch, J., Ward, K., Smith, B., Levy, M., Cummings, M.D., Haltiwanger, R.C., Trescher, G., Wang, B., Hemling, M.E., Quinn, C.J., Cheng, H.-Y., Lin, F., Smith, W.W., Janson, C.A., Zhao, B., McQueney, M.S., D'Alessio, K., Lee, C.P., Marzulli, A., Dodds, R.A., Blake, S., Hwang, S.M., James, I.E., Gress, C.J., Bradley, B.R., Lark, M.W., Gowen, M., Veber, D.F.
J.Med.Chem.
HeaderHydrolase
Released2003-01-07
Resolution2.400
CATH Insert Date05 Mar, 2006

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
1nljA00 05 Mar, 2006 3.90.70.10 Assigned
1nljB00 05 Mar, 2006 3.90.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P43235 CATK_HUMAN Homo sapiens Cathepsin K
P43235 CATK_HUMAN Homo sapiens Cathepsin K