PDB Information

PDB1MTR
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 1
Primary Citation
Substrate-based cyclic peptidomimetics of Phe-Ile-Val that inhibit HIV-1 protease using a novel enzyme-binding mode.
March, D.R., Abbenante, G., Bergman, D.A., Brinkworth, R.I., Wickramasinghe, W., Begun, J., Martin, J.L., Fairlie, D.P.
J.Am.Chem.Soc.
HeaderHydrolase/Hydrolase Inhibitor
Released1996-02-15
Resolution1.750
CATH Insert Date05 Mar, 2006

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
1mtrA00 05 Mar, 2006 2.40.70.10 Assigned
1mtrB00 05 Mar, 2006 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P03369 POL_HV1A2 HIV-1 M:B_ARV2/SF2 Gag-Pol polyprotein
P03369 POL_HV1A2 HIV-1 M:B_ARV2/SF2 Gag-Pol polyprotein