PDB Information

PDB1LPG
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Design and Quantitative Structure-Activity relationship of 3-amidinobenzyl-1H-indole-2-carboxamides as potent, nonchiral, and selective inhibitors of blood coagulation factor Xa.
Matter, H., Defossa, E., Heinelt, U., Blohm, P.M., Schneider, D., Mueller, A., Herok, S., Schreuder, H., Liesum, A., Brachvogel, B., Loenze, P., Walser, A., Al-Obeidi, F., Wildgoose, P.
J.Med.Chem.
HeaderHydrolase
Released2002-05-08
Resolution2.000
CATH Insert Date05 Mar, 2006

PDB Images (6)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
1lpgA00 05 Mar, 2006 2.10.25.10 Assigned
1lpgB01 05 Mar, 2006 2.40.10.10 Assigned
1lpgB02 05 Mar, 2006 2.40.10.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00742 FA10_HUMAN Homo sapiens Coagulation factor X
P00742 FA10_HUMAN Homo sapiens Coagulation factor X