PDB Information

PDB1H1R
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Structure-based design of a potent purine-based cyclin-dependent kinase inhibitor.
Davies, T.G., Bentley, J., Arris, C.E., Boyle, F.T., Curtin, N.J., Endicott, J.A., Gibson, A.E., Golding, B.T., Griffin, R.J., Hardcastle, I.R., Jewsbury, P., Johnson, L.N., Mesguiche, V., Newell, D.R., Noble, M.E., Tucker, J.A., Wang, L., Whitfield, H.J.
Nat. Struct. Biol.
HeaderTransferase
Released2002-07-21
Resolution2.000
CATH Insert Date05 Mar, 2006

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped
C 05 Mar, 2006 Chopped
D 05 Mar, 2006 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
1h1rA01 05 Mar, 2006 3.30.200.20 Assigned
1h1rA02 05 Mar, 2006 1.10.510.10 Assigned
1h1rB01 05 Mar, 2006 1.10.472.10 Assigned
1h1rB02 05 Mar, 2006 1.10.472.10 Assigned
1h1rC01 05 Mar, 2006 3.30.200.20 Assigned
1h1rC02 05 Mar, 2006 1.10.510.10 Assigned
1h1rD01 05 Mar, 2006 1.10.472.10 Assigned
1h1rD02 05 Mar, 2006 1.10.472.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2
P20248 CCNA2_HUMAN Homo sapiens Cyclin-A2