CATH Classification

Domain Context

CATH Clusters

Superfamily Cyclin-like
Functional Family G2/mitotic-specific cyclin-B1

Enzyme Information

UniProtKB Entries (1)

P06493
CDK1_HUMAN
Homo sapiens
Cyclin-dependent kinase 1

PDB Structure

PDB 5LQF
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Cyclin-Dependent Kinase (CDK) Inhibitors: Structure-Activity Relationships and Insights into the CDK-2 Selectivity of 6-Substituted 2-Arylaminopurines.
Coxon, C.R., Anscombe, E., Harnor, S.J., Martin, M.P., Carbain, B., Golding, B.T., Hardcastle, I.R., Harlow, L.K., Korolchuk, S., Matheson, C.J., Newell, D.R., Noble, M.E., Sivaprakasam, M., Tudhope, S.J., Turner, D.M., Wang, L.Z., Wedge, S.R., Wong, C., Griffin, R.J., Endicott, J.A., Cano, C.
J. Med. Chem.