CATH Classification

Domain Context

CATH Clusters

Superfamily Cyclin-like
Functional Family Putative cyclin-c

Enzyme Information

UniProtKB Entries (1)

P49336
CDK8_HUMAN
Homo sapiens
Cyclin-dependent kinase 8

PDB Structure

PDB 5IDN
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Structure-Based Optimization of Potent, Selective, and Orally Bioavailable CDK8 Inhibitors Discovered by High-Throughput Screening.
Czodrowski, P., Mallinger, A., Wienke, D., Esdar, C., Poschke, O., Busch, M., Rohdich, F., Eccles, S.A., Ortiz-Ruiz, M.J., Schneider, R., Raynaud, F.I., Clarke, P.A., Musil, D., Schwarz, D., Dale, T., Urbahns, K., Blagg, J., Schiemann, K.
J. Med. Chem.