CATH Classification

Domain Context

CATH Clusters

Superfamily YVTN repeat-like/Quinoprotein amine dehydrogenase
Functional Family WD repeat-containing protein 5

Enzyme Information

UniProtKB Entries (1)

P61964
WDR5_HUMAN
Homo sapiens
WD repeat-containing protein 5

PDB Structure

PDB 5EAM
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Structure-Based Optimization of a Small Molecule Antagonist of the Interaction Between WD Repeat-Containing Protein 5 (WDR5) and Mixed-Lineage Leukemia 1 (MLL1).
Getlik, M., Smil, D., Zepeda-Velazquez, C., Bolshan, Y., Poda, G., Wu, H., Dong, A., Kuznetsova, E., Marcellus, R., Senisterra, G., Dombrovski, L., Hajian, T., Kiyota, T., Schapira, M., Arrowsmith, C.H., Brown, P.J., Vedadi, M., Al-Awar, R.
J. Med. Chem.