CATH Classification

Domain Context

CATH Clusters

Superfamily YVTN repeat-like/Quinoprotein amine dehydrogenase
Functional Family WD repeat-containing protein 5

Enzyme Information

UniProtKB Entries (1)

P61964
WDR5_HUMAN
Homo sapiens
WD repeat-containing protein 5

PDB Structure

PDB 4IA9
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Synthesis, Optimization, and Evaluation of Novel Small Molecules as Antagonists of WDR5-MLL Interaction.
Bolshan, Y., Getlik, M., Kuznetsova, E., Wasney, G.A., Hajian, T., Poda, G., Nguyen, K.T., Wu, H., Dombrovski, L., Dong, A., Senisterra, G., Schapira, M., Arrowsmith, C.H., Brown, P.J., Al-Awar, R., Vedadi, M., Smil, D.
ACS Med Chem Lett