CATH Classification

Domain Context

CATH Clusters

Superfamily SET domain
Functional Family Histone-lysine N-methyltransferase

Enzyme Information

2.1.1.-
Methyltransferases.
based on mapping to UniProt Q9BYW2
2.1.1.43
Histone-lysine N-methyltransferase.
based on mapping to UniProt Q9BYW2
S-adenosyl-L-methionine + L-lysine-[histone] = S-adenosyl-L-homocysteine + N(6)-methyl-L-lysine-[histone].

UniProtKB Entries (1)

Q9BYW2
SETD2_HUMAN
Homo sapiens
Histone-lysine N-methyltransferase SETD2

PDB Structure

PDB 4H12
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Sinefungin Derivatives as Inhibitors and Structure Probes of Protein Lysine Methyltransferase SETD2.
Zheng, W., Ibanez, G., Wu, H., Blum, G., Zeng, H., Dong, A., Li, F., Hajian, T., Allali-Hassani, A., Amaya, M.F., Siarheyeva, A., Yu, W., Brown, P.J., Schapira, M., Vedadi, M., Min, J., Luo, M.
J.Am.Chem.Soc.