CATH Classification

Domain Context

CATH Clusters

Superfamily Bromodomain-like
Functional Family Bromodomain-containing protein 4

Enzyme Information

UniProtKB Entries (1)

O60885
BRD4_HUMAN
Homo sapiens
Bromodomain-containing protein 4

PDB Structure

PDB 4A9L
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Fragment-Based Discovery of Bromodomain Inhibitors Part 1: Inhibitor Binding Modes and Implications for Lead Discovery.
Chung, C.W., Dean, A.W., Woolven, J.M., Bamborough, P.
J.Med.Chem.